1960 　R. B. Woodward
1962 　John D. Roberts
1963 　M. S. Newman
1964 　Saul Winstein
1965 　Ronald Breslow
1966 　Gilbert Stork
1967 　George H. Buchi
1968 　Emmanuel Vogel
1969 　Frank H. Westheimer
1970 　Albert Eschenmoser
1971 　Michael J. S. Dewar
1971 　Paul Bartlett
1973 　Duilio Arigoni
1974 　Rolf Huisgen
1975 　Jean-Marie Lehn
1976 　Gunther Wilke
1978 　H. E. Simmons
1979 　Teruaki Mukaiyama
1980 　Jack Baldwin
1982 　Alan R. Battersby, F.R.S.
1983 　Martin Saunders
1984 　Josef Michl
1985 　Jeremy R. Knowles
1986 　Dieter Seebach
1987 　Sir Derek Barton
1988 　Peter B. Dervan
1989 　Kurt Mislow
1990 　A.L.J. Beckwith, FAA, FRS
1991 　Ryoji Noyori
1992 　Manfred T. Reetz
1993 　John T. Groves
1994 　Kyriacos Nicolaou
1996 　Jean M.J. Fréchet
1997 　Mary Anne Fox
1998 　Jean-Pierre Sauvage
1999 　Guy Bertrand
2000 　Dennis Dougherty
2000 　Hisashi Yamamoto
2003 　Barry Trost
2005 　William Degrado
2006 　Tamio Hayashi
2007 　B. L. (Ben) Feringa
2008 　Daniel Kahne
2009 　JoAnne Stubbe
2011 　David MacMillan
2012 　Makoto Fujita